A β-adrenergic receptor agonist that putatively through activation of protein kinase A increases protein synthesis in skeletal muscle fibers

Zilpaterol (hydrochloride) – 1 mg

Brand:
Cayman
CAS:
119520-06-8
Storage:
-20
UN-No:
Non-Hazardous - /

Zilpaterol is a β-adrenergic receptor agonist that putatively through activation of protein kinase A increases protein synthesis in skeletal muscle fibers, as well as reduces lipogenesis and increases lipolysis in adipose tissues.{26935,26936} It was approved by the FDA in 2006 as a veterinary food additive for the purpose of increasing lean body weight and improving feed efficiency in commercial beef cattle.{26937}  

 

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Description

A β-adrenergic receptor agonist that putatively through activation of protein kinase A increases protein synthesis in skeletal muscle fibers, as well as reduces lipogenesis and increases lipolysis in adipose tissues; used as a veterinary food additive to increase lean body weight in commercial beef cattle

Formal name: (6R,7R)-rel-4,5,6,7-tetrahydro-7-hydroxy-6-[(1-methylethyl)amino]-imidazo[4,5,1-jk][1]benzazepin-2(1H)-one, monohydrochloride

Synonyms:  RU-42173

Molecular weight: 297.8

CAS: 119520-06-8

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Endocrinology & Metabolism|Cofactors & Vitamins

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