A major phase I metabolite of the mycotoxin α-zearalanol (zeranol)

Zearalanone – 5 mg

Brand:
Cayman
CAS:
5975-78-0
Storage:
-20
UN-No:
Non-Hazardous - /

Zearalanone is a major phase I metabolite of the mycotoxin α-zearalanol (zeranol), a non-steroidal estrogen produced by fungi.{31431,31433} Zearalanone is an estrogen receptor agonist (EC50 = 0.11 µM).{31432} It also acts as an androgen receptor antagonist.{31434} Zearalanone, zearalenone (Item No. 11353), and related compounds can be abundant in plant material infected with Fusarium.{31430}  

 

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Description

A major phase I metabolite of the mycotoxin α-zearalanol (zeranol), a non-steroidal estrogen produced by fungi; an estrogen receptor agonist (EC50 = 0.11 µM)

Formal name: (3S)-3,4,5,6,9,10,11,12-octahydro-14,16-dihydroxy-3-methyl-1H-2-benzoxacyclotetradecin-1,7(8H)-dione

Synonyms: 

Molecular weight: 320.4

CAS: 5975-78-0

Purity: ≥98%

Formulation: A crystalline solid

Application|Mass Spectrometry||Product Type|Biochemicals|Receptor Pharmacology|Agonists||Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Product Type|Biochemicals|Toxins|Mycotoxins||Product Type|Biochemicals|Xenobiotic Metabolites||Research Area|Endocrinology & Metabolism|Hormones & Receptors|Androgens||Research Area|Endocrinology & Metabolism|Hormones & Receptors|Estrogens & Progestins

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