A selective 5-HT6 receptor agonist (EC50 = 7.3 nM at the human 5-HT6 receptor); increases cortical GABA levels in rat frontal cortex

WAY-208466 (hydrochloride) – 1 mg

Brand:
Cayman
CAS:
1207064-61-6
Storage:
-20
UN-No:
Non-Hazardous - /

WAY-208466 is a selective 5-HT6 receptor agonist (EC50 = 7.3 nM at the human 5-HT6 receptor).{32648} It has been shown to increase cortical GABA levels in rat frontal cortex, producing anxiolytic-like effects in vivo. {32648}  

 

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SKU: 11938 - 1 mg Category:

Description

A selective 5-HT6 receptor agonist (EC50 = 7.3 nM at the human 5-HT6 receptor); increases cortical GABA levels in rat frontal cortex, producing anxiolytic-like effects in vivo

Formal name: 3-[(3-fluorophenyl)sulfonyl]-N,N-dimethyl-1H-pyrrolo[2,3-b]pyridine-1-ethanamine, dihydrochloride

Synonyms: 

Molecular weight: 420.3

CAS: 1207064-61-6

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Neuroscience|Behavioral Neuroscience|Anxiety

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