A major metabolite of voriconazole; formed via oxidation of voriconazole by CYP3A4 and CYP2C19

Voriconazole N-oxide – 10 mg

Brand:
Cayman
CAS:
618109-05-0
Storage:
-20
UN-No:
- 2811 / 6.1

Voriconazole N-oxide is a major metabolite of the triazole antifungal voriconazole (Item No. 15633).{48321} It is formed via oxidation of voriconazole by the cytochrome P450 (CYP) isoforms CYP3A4 and CYP2C19.  

 

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SKU: 28047 - 10 mg Category:

Description

A major metabolite of voriconazole; formed via oxidation of voriconazole by CYP3A4 and CYP2C19

Formal name: (αR,βS)-α-(2,4-difluorophenyl)-5-fluoro-β-methyl-α-(1H-1,2,4-triazol-1-ylmethyl)-4-pyrimidineethanol, 1-oxide

Synonyms:  UK 121265

Molecular weight: 365.3

CAS: 618109-05-0

Purity: ≥95%

Formulation: A solid

Product Type|Biochemicals|Xenobiotic Metabolites||Research Area|Immunology & Inflammation||Research Area|Infectious Disease|Fungal Diseases|Aspergillosis||Research Area|Infectious Disease|Fungal Diseases|Candidiasis||Research Area|Toxicology|Drug Metabolism|Cytochrome P450||Research Area|Toxicology|Drug Metabolism|Drug Metabolites

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