A neonicotinoid insecticide; acts as a selective agonist at insect nAChRs (IC50s = 2.7 and 860 nM for Drosophila nAChRs and M10 mouse fibroblast cells expressing α4β2 subunit-containing nAChRs

Thiacloprid – 50 mg

Brand:
Cayman
CAS:
111988-49-9
Storage:
-20
UN-No:
De Minimis - 2811 / 6.1

Thiacloprid is a neonicotinoid insecticide that acts as a selective agonist at insect nicotinic acetylcholine receptors (nAChRs) with IC50 values of 2.7 and 860 nM for Drosophila nAChRs and M10 mouse fibroblast cells expressing α4β2 subunit-containing nAChRs, respectively.{33400} It is active against aphids, whiteflies, various species of beetle, and Lepidoptera species when used at concentrations ranging from 48 to 180 g AI/hectare.{45005} It has anti-estrogenic activity in a yeast estrogen screen and is toxic to adult female houseflies and mice (LD50s = 0.03 and 28 mg/kg, respectively).{33400,45006} Formulations containing thiacloprid have been used in the control of insects in agriculture.  

 

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Description

A neonicotinoid insecticide; acts as a selective agonist at insect nAChRs (IC50s = 2.7 and 860 nM for Drosophila nAChRs and M10 mouse fibroblast cells expressing α4β2 subunit-containing nAChRs, respectively); active against aphids, whiteflies, various species of beetle, and Lepidoptera species at 48-180 g AI/hectare; has anti-estrogenic activity in a yeast estrogen screen; toxic to adult female houseflies and mice (LD50s = 0.03 and 28 mg/kg, respectively)

Formal name: [N(Z)]-N-[3-[(6-chloro-3-pyridinyl)methyl]-2-thiazolidinylidene]-cyanamide

Synonyms:  BAY YRC 2894

Molecular weight: 252.7

CAS: 111988-49-9

Purity: ≥98%

Formulation: A solid

Product Type|Biochemicals|Ion Channel Modulation|Activators||Product Type|Biochemicals|Pesticides|Insecticides||Research Area|Toxicology|Environmental|Agriculture||Research Area|Toxicology|Environmental|Endocrine Disruption

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