A small molecule activator of p53; increases p53 activity in MCF-7 cells at 10 µM; increases the level of K40-acetylated α-tubulin in H1299 cells; inhibits SIRT2 protein deacetylase activity

Tenovin-3 – 1 mg

Brand:
Cayman
CAS:
1011301-27-1
Storage:
-20
UN-No:
Non-Hazardous - /

Tenovin-3 is a small molecule activator of p53 transcriptional activity.{16243} It increases p53 activity in MCF-7 cells when used at a concentration of 10 µM. It also increases the level of K40-acetylated α-tubulin in H1299 cells and inhibits SIRT2 protein deacetylase activity.  

 

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Description

A small molecule activator of p53; increases p53 activity in MCF-7 cells at 10 µM; increases the level of K40-acetylated α-tubulin in H1299 cells; inhibits SIRT2 protein deacetylase activity

Formal name: N-[[(4-aminophenyl)amino]thioxomethyl]-4-(1,1-dimethylethyl)-benzamide

Synonyms: 

Molecular weight: 327.4

CAS: 1011301-27-1

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Small Molecule Activators|Transcription Factors & Coactivators||Research Area|Epigenetics, Transcription, & Translation|Erasers|Histone Deacetylation||Research Area|Epigenetics, Transcription, & Translation|Transcription Factors

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