A major metabolite of telmisartan; does not bind human serum albumin; is cleared from rat plasma with a clearance rate of 180 ml/min/kg following intravenous administration

Telmisartan Acyl-β-D-Glucuronide – 1 mg

Brand:
Cayman
CAS:
250780-40-6
Storage:
-20
UN-No:
Non-Hazardous - /

Telmisartan acyl-β-D-glucuronide is a major metabolite of the angiotensin II receptor antagonist telmisartan (Item No. 11615).{48353} It does not bind human serum albumin and is cleared from rat plasma with a clearance rate of 180 ml/min/kg following intravenous administration.  

 

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SKU: 28056 - 1 mg Category:

Description

A major metabolite of telmisartan; does not bind human serum albumin; is cleared from rat plasma with a clearance rate of 180 ml/min/kg following intravenous administration

Formal name: 1-[4′-[(1,4′-dimethyl-2′-propyl[2,6′-bi-1H-benzimidazol]-1′-yl)methyl][1,1′-biphenyl]-2-carboxylate] β-D-glucopyranuronic acid

Synonyms:  Telmisartan Glucuronide

Molecular weight: 690.7

CAS: 250780-40-6

Purity: ≥95%

Formulation: A solid

Product Type|Biochemicals|Xenobiotic Metabolites||Research Area|Cardiovascular System|Cardiovascular Diseases|Hypertension||Research Area|Cardiovascular System|Heart|Myocardial Hypertrophy||Research Area|Cardiovascular System|Kidney & Renal Disease||Research Area|Toxicology|Drug Metabolism|Drug Metabolites

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