A selective α2-adrenoceptor antagonist that shows nanomolar Ki values for the three subtypes

SKF 86466 (hydrochloride) – 1 mg

Brand:
Cayman
CAS:
86129-54-6
Storage:
-20
UN-No:
Non-Hazardous - /

SKF 86466 is a selective antagonist of α2-adrenoceptors that shows nanomolar Ki values for the three subtypes, α2A, α2B, and α2C.{34495,34497} It is active in vivo, evoking antihypertensive effects in animal studies and clinical trials.{34494,34497} SKF 86466 is used to study the role of α2-adrenoceptors in animals.{34496,34498}  

 

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SKU: 11953 - 1 mg Category:

Description

A selective α2-adrenoceptor antagonist that shows nanomolar Ki values for the three subtypes, α2A, α2B, and α2C; evokes antihypertensive effects in animal studies and clinical trials

Formal name: 6-chloro-2,3,4,5-tetrahydro-3-methyl-1H-3-benzazepine, monohydrochloride

Synonyms: 

Molecular weight: 232.2

CAS: 86129-54-6

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Cardiovascular System|Cardiovascular Diseases|Hypertension

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