A polymethoxylated flavone that has been shown to enhance adipogenesis and lipolysis

Sinensetin – 5 mg

Brand:
Cayman
CAS:
2306-27-6
Storage:
-20
UN-No:
De Minimis - 2811 / 6.1

Sinensetin is a polymethoxylated flavone that is present in the Southeast Asian medical plant O. stamineus, as well as in orange oil. It has been shown to enhance adipogenesis and lipolysis by increasing cAMP levels in 3T3-L1 cells.{31727} Sinensetin is also reported to inhibit α-glucosidase and α-amylase activity in vitro, indicating its potential usefulness in the control of glucose absorption.{31728} Additionally, sinensetin has been shown to suppress the expression of genes associated with inflammation by regulating IκBα protein levels in LPS-activated macrophages.{31729}  

 

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Description

A polymethoxylated flavone that has been shown to enhance adipogenesis and lipolysis, to inhibit α-glucosidase and α-amylase activity, and to suppress the expression of genes associated with inflammation by regulating IκBα

Formal name: 2-(3,4-dimethoxyphenyl)-5,6,7-trimethoxy-4H-1-benzopyran-4-one

Synonyms:  Pedalitin Permethyl ether

Molecular weight: 372.4

CAS: 2306-27-6

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Natural Products|Flavonoids||Product Type|Biochemicals|Small Molecule Inhibitors|MMPs||Research Area|Endocrinology & Metabolism|Carbohydrate Metabolism||Research Area|Endocrinology & Metabolism|Metabolic Diseases|Obesity||Research Area|Immunology & Inflammation|Innate Immunity

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