A potent

Senktide – 5 mg

Brand:
Cayman
CAS:
106128-89-6
Storage:
-20
UN-No:
Non-Hazardous - /

Senktide is a potent, selective agonist of the neuromedin K3 (NK3) receptor (EC50 = 0.5-3 nM).{28054,28052,28050} It less potently agonizes the NK1 receptor (EC50 = 35 µM) and is without effect on the NK2 receptor.{28054,28052,28050} Senktide is used to study the action of the NK3 receptor in cells and in animals.{28051,28053}  

 

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Description

A potent, selective agonist of the neuromedin K3 (NK3) receptor (EC50 = 0.5-3 nM); used to study the action of the NK3 receptor in cells and in animals

Formal name: N-(3-carboxy-1-oxopropyl)-L-α-aspartyl-L-phenylalanyl-N-methyl-L-phenylalanylglycyl-L-leucyl-L-methioninamide

Synonyms: 

Molecular weight: 842

CAS: 106128-89-6

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Endocrinology & Metabolism|Hormones & Receptors||Research Area|Neuroscience

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