An MMP inhibitor (IC50s = 50s = >10

SD 2590 (hydrochloride) – 5 mg

Brand:
Cayman
CAS:
226395-93-3
Storage:
-20
UN-No:
Non-Hazardous - /

SD 2590 is an inhibitor of matrix metalloproteinase-2 (MMP-2), -3, -8, -9, and -13 (IC50s = 50s = >10,000 and 7,000 nM, respectively). SD 2590 (10 mg/kg per day) inhibits dilation of the left ventricle in rats following myocardial infarction (MI) compared to MI vehicle control animals.  

 

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SKU: 27680 - 5 mg Category:

Description

An MMP inhibitor (IC50s = 50s = >10,000 and 7,000 nM, respectively); inhibits dilation of the left ventricle in rats following MI compared to MI vehicle control animals at 10 mg/kg per day.

Formal name: N-hydroxy-1-(2-methoxyethyl)-4-[[4-[4-(trifluoromethoxy)phenoxy]phenyl]sulfonyl]-4-piperidinecarboxamide, monohydrochloride

Synonyms:  SC-78080

Molecular weight: 555

CAS: 226395-93-3

Purity: ≥98%

Formulation: A solid

Product Type|Biochemicals|Small Molecule Inhibitors|MMPs||Research Area|Cardiovascular System|Cardiovascular Diseases|Myocardial Infarction||Research Area|Cell Biology|Proteolysis|Cytosolic & Secreted Proteases

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