A β2-AR agonist; induces relaxation of isolated pig detrusor muscle from 0.001-1 μM; reduces electrically-induced isometric tension in myometrial strips isolated from rabbits on day 25 of pregnancy at 30 μg/ml; suppresses spontaneous motility of and increases concentration of cAMP in isolated pregnant rat uterus

Ritodrine (hydrochloride) – 500 mg

Brand:
Cayman
CAS:
23239-51-2
Storage:
-20
UN-No:
Non-Hazardous - /

Ritodrine is an agonist of β2-adrenergic receptors (β2-ARs).{47089} It induces relaxation of isolated pig detrusor muscle when used at concentrations ranging from 0.001 to 1 μM. Ritodrine (30 μg/ml) reduces electrically-induced isometric tension in myometrial strips isolated from rabbits on day 25 of pregnancy.{47090} It also suppresses spontaneous motility of and increases concentration of cyclic AMP (cAMP) in isolated pregnant rat uterus.{47091} Formulations containing ritodrine were previously used to stop premature labor.  

 

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SKU: 26084 - 500 mg Category:

Description

A β2-AR agonist; induces relaxation of isolated pig detrusor muscle from 0.001-1 μM; reduces electrically-induced isometric tension in myometrial strips isolated from rabbits on day 25 of pregnancy at 30 μg/ml; suppresses spontaneous motility of and increases concentration of cAMP in isolated pregnant rat uterus

Formal name: (αS)-rel-4-hydroxy-α-[(1R)-1-[[2-(4-hydroxyphenyl)ethyl]amino]ethyl]-benzenemethanol, monohydrochloride

Synonyms:  (±)-Ritodrine|DU 21220|NSC 291565

Molecular weight: 323.8

CAS: 23239-51-2

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Endocrinology & Metabolism|Reproductive Biology

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