A derivative of ketanserin in which the 4-(p-fluorobenzoyl)piperidine group has been replaced with an N-(2-methoxybenzyl) moiety

RH-34 – 10 mg

Brand:
Cayman
CAS:
1028307-48-3
Storage:
-20
UN-No:
Non-Hazardous - /

Ketanserin is a potent antagonist of the serotonin receptor 5-HT2A (Ki = 3.16 nM) that has hypertensive effects in vivo.{26494,26493} RH-34 is a derivative of ketanserin in which the 4-(p-fluorobenzoyl)piperidine group has been replaced with an N-(2-methoxybenzyl) moiety. In phenethylamines, which are 5-HT2A agonists, this addition increases the affinity and selectivity for the 5-HT2A receptor over other serotonin receptors.{20442} The physiological and toxicological properties of this compound are not known. This product is intended for forensic and research applications.  

 

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Description

A derivative of ketanserin in which the 4-(p-fluorobenzoyl)piperidine group has been replaced with an N-(2-methoxybenzyl) moiety

Formal name: 3-[2-[[(2-methoxyphenyl)methyl]amino]ethyl]-2,4(1H,3H)-quinazolinedione

Synonyms: 

Molecular weight: 325.4

CAS: 1028307-48-3

Purity: ≥95%

Formulation: A crystalline solid

Application|Mass Spectrometry||Product Type|Biochemicals|Analytical Standards||Research Area|Forensic Chemistry & Toxicology|Hallucinogens|Phenethylamines||Research Area|Forensic Chemistry & Toxicology|Stimulants|Phenethylamines

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