A selective

Regadenoson – 10 mg

Brand:
Cayman
CAS:
313348-27-5
Storage:
-20
UN-No:
Non-Hazardous - /

Regadenoson is a selective, short-acting adenosine A2A receptor agonist (Ki = 1.1 nM for pig striatum A2A receptor).{30539,30542} It increases coronary blood flow 3.4- to 3.8-fold with a half-time to reversal of 1.9-2.6 minutes in open-chest anesthetized pigs.{30539} Regadenoson is used to induce hyperemia (increased blood flow), particularly in the context of myocardial perfusion imaging.{30537,30541} It has also been found to increase the delivery of compounds to the central nervous system through the blood-brain barrier in animals.{30538,30540}  

 

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Description

A selective, short-acting adenosine A2A receptor agonist (Ki = 1.1 nM for pig striatum A2A receptor); used to induce hyperemia, particularly in the context of myocardial perfusion imaging

Formal name: 2-[4-[(methylamino)carbonyl]-1H-pyrazol-1-yl]-adenosine

Synonyms:  CVT-3146|Lexiscan

Molecular weight: 390.4

CAS: 313348-27-5

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Cardiovascular System|Vasculature|Vasodilation||Research Area|Neuroscience

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