An orally bioavailable SARM that binds to the androgen receptor with a Ki value of 7 nM; stimulates muscle weight increase without affecting prostate or seminal vesicle in castrated male rats

RAD140 – 500 µg

Brand:
Cayman
CAS:
1182367-47-0
Storage:
-20
UN-No:
Non-Hazardous - /

RAD140 is an orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM) that binds to the androgen receptor with a Ki value of 7 nM.{32428} At 0.03-0.3 mg/kg, it has been shown to stimulate muscle weight increase without affecting prostate or seminal vesicle in castrated male rats.{32428} At 0.3-1 mg/kg, RAD140 demonstrates partial antagonist activity in seminal vesicle and prostate.{32428}  

 

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Description

An orally bioavailable SARM that binds to the androgen receptor with a Ki value of 7 nM; stimulates muscle weight increase without affecting prostate or seminal vesicle in castrated male rats

Formal name: 2-chloro-4-[[(1R,2S)-1-[5-(4-cyanophenyl)-1,3,4-oxadiazol-2-yl]-2-hydroxypropyl]amino]-3-methyl-benzonitrile

Synonyms:  Testolone

Molecular weight: 393.8

CAS: 1182367-47-0

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Endocrinology & Metabolism|Hormones & Receptors|Androgens

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