A selective dopamine D2/D3 receptor antagonist (Kis = 1.8

Raclopride – 25 mg

Brand:
Cayman
CAS:
84225-95-6
Storage:
-20
UN-No:
Non-Hazardous - /

Raclopride is a selective dopamine D2/D3 receptor antagonist with Ki values of 1.8, 3.5, 2,400, and 18,000 nM for D2, D3, D4, and D1 receptors, respectively.{32473} It passes the blood brain barrier and can be used in in vivo binding and autoradiography studies of the dopamine system under normal and pathological conditions such as Huntington’s disease.{32472,32471}  

 

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Description

A selective dopamine D2/D3 receptor antagonist (Kis = 1.8, 3.5, 2,400, and 18,000 nM for D2, D3, D4, and D1 receptors, respectively); used in in vivo binding and autoradiography studies of the dopamine system

Formal name: 3,5-dichloro-N-[[(2S)-1-ethyl-2-pyrrolidinyl]methyl]-2-hydroxy-6-methoxy-benzamide

Synonyms:  (S)-(-)-Raclopride

Molecular weight: 347.2

CAS: 84225-95-6

Purity: ≥98%

Formulation: A solid

Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Neuroscience|Neurodegenerative Disorders|Huntington’s Disease

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