A selective

R-(−)-Deprenyl (hydrochloride) – 500 mg

Brand:
Cayman
CAS:
14611-52-0
Storage:
-20
UN-No:
Non-Hazardous - /

Monoamine oxidase (MAO) inhibitors have utility in ameliorating a variety of neurological conditions, including depression.{23885} R-(−)-Deprenyl is a selective, reversible inhibitor of MAO-B (Ki = 0.091 μM) over MAO-A (Ki = 9.06 μM).{23886,23884} In addition to finding use against depression, R-(−)-deprenyl provides neuroprotection which may be relevant to Parkinson’s disease, Alzheimer’s disease, Huntington’s disease, and stroke.{15160,23885} The ability of this compound to slow the progression of disability in early Parkinson’s disease may be independent of its effects on MAO activity.{15160}  

 

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Description

A selective, reversible inhibitor of MAO-B (Ki = 0.091 μM) over MAO-A (Ki = 9.06 μM); may ameliorate depression, Parkinson’s disease, Alzheimer’s disease, Huntington’s disease, and stroke

Formal name: (R)-N,α-dimethyl-N-2-propyn-1-yl-benzeneethanamine, monohydrochloride

Synonyms:  L-Deprenyl|Selegiline

Molecular weight: 223.7

CAS: 14611-52-0

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Small Molecule Inhibitors||Research Area|Neuroscience|Neurodegenerative Disorders|Alzheimer’s Disease||Research Area|Neuroscience|Neurodegenerative Disorders|Parkinson’s Disease

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