2-AG exhibits CB agonist activity at the CB1 receptor

Prostaglandin F2α serinol amide – 5 mg

Brand:
Cayman
CAS:
1135226-99-1
Storage:
-20
UN-No:
De Minimis - 1170 / 3

2-Arachidonyl glycerol (2-AG) exhibits cannabinoid agonist activity at the CB1 receptor,{5306} is an important endogenous monoglyceride species,{6819} and is thus considered to be the natural ligand for the CB1 receptor. 2-AG can also be metabolized by COX-2 and prostaglandin D, E, F, and I synthases to form prostaglandin 2-glyceryl (PG 2-glyceryl) esters.{11045} PGF2α-SA is a stable analog of PGF2α 2-glyceryl ester. The biological activity of PGF2α-SA has not yet been determined.  

 

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SKU: 10194 - 5 mg Category:

Description

2-AG exhibits CB agonist activity at the CB1 receptor,{5306} is an important endogenous monoglyceride species,{6819} and is thus considered to be the natural ligand for the CB1 receptor. 2-AG can also be metabolized by COX-2 and PGD, E, F, and I synthases to form PG 2-glyceryl esters.{11045} PGF2α-SA is a stable analog of PGF2α 2-glyceryl ester. The biological activity of PGF2α-SA has not yet been determined.

Formal name: N-[(2-hydroxy-1-hydroxymethyl)ethyl]-9α,11α,15S-trihydroxy-prosta-5Z,13E-dien-1-amide

Synonyms:  PGF2α-SA

Molecular weight: 427.6

CAS: 1135226-99-1

Purity: ≥98%

Formulation: A solution in ethanol

Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway||Research Area|Lipid Biochemistry|Endocannabinoid/Endocannabinoid-like||Research Area|Neuroscience|Cannabinoid Research

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