PGF2α dimethyl amine is a derivative of PGF2α which was designed as a PG antagonist for in vitro and in vivo studies.{1319} PGF2α dimethyl amine is a weak FP receptor antagonist.{1319} In gerbil colon

Prostaglandin F2α dimethyl amine – 1 mg

Brand:
Cayman
CAS:
67508-09-2
Storage:
-20
UN-No:
De Minimis - 1170 / 3

PGF2α dimethyl amine is a derivative of PGF2α which was designed as a PG antagonist for in vitro and in vivo studies.{1319} PGF2α dimethyl amine is a weak FP receptor antagonist.{1319} In gerbil colon, PGF2α dimethyl amine at a dose of 3.2 µg/ml inhibits the contractile effects of PGF2α (at 6 ng/ml) by 60%.{1319}  

 

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Description

PGF2α dimethyl amine is a derivative of PGF2α which was designed as a PG antagonist for in vitro and in vivo studies.{1319} PGF2α dimethyl amine is a weak FP receptor antagonist.{1319} In gerbil colon, PGF2α dimethyl amine at a dose of 3.2 µg/ml inhibits the contractile effects of PGF2α (at 6 ng/ml) by 60%.{1319}

Formal name: N,N,-dimethyl-9α,11α,15S-trihydroxy-prosta-5Z,13E-dien-1-amine

Synonyms:  Dinoprost dimethyl amine|PGF2α dimethyl amine

Molecular weight: 367.6

CAS: 67508-09-2

Purity: ≥98%

Formulation: A solution in ethanol

Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway

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