A PCKζ inhibitor; 8

PKC-9 – 5 mg

Brand:
Cayman
CAS:
1132609-87-0
Storage:
-20
UN-No:
Non-Hazardous - /

PKC-9 is an inhibitor of PKCζ that is 8,000-, 20,671-, 711-, 918-, 1,895-, 12,424-, 10-, and 1,218-fold selective for PKCζ over PKCα, PKCβII, PKCγ, PKCδ, PKCε, PKCη, PKCι, and PKCθ, respectively.{36787} It also inhibits 27 additional kinases in a panel of 37 kinases when used at a concentration of 10 μM.  

 

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SKU: 25556 - 5 mg Category:

Description

A PCKζ inhibitor; 8,000-, 20,671-, 711-, 918-, 1,895-, 12,424-, 10-, and 1,218-fold selective for PKCζ over PKCα, PKCβII, PKCγ, PKCδ, PKCε, PKCη, PKCι, and PKCθ, respectively; inhibits 27 additional kinases in a panel of 37 kinases at 10 μM

Formal name: 4-[3-[7-(4-methyl-1-piperazinyl)-1H-benzimidazol-2-yl]-1H-indazol-6-yl]-benzenamine

Synonyms: 

Molecular weight: 423.5

CAS: 1132609-87-0

Purity: ≥95%

Formulation: A solid

Product Type|Biochemicals|Kinase Inhibitors|PKC||Product Type|Biochemicals|Small Molecule Inhibitors|Kinases||Research Area|Cell Biology|Cell Signaling

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