An antispasmodic agent; an inhibitor of AChE (Kis = 36 and 45 μM for bovine erythrocyte and electric eel enzyme

Pitofenone (hydrochloride) – 50 mg

Brand:
Cayman
CAS:
1248-42-6
Storage:
-20
UN-No:
Non-Hazardous - /

Pitofenone is an antispasmodic agent and an inhibitor of acetylcholinesterase (AChE; Kis = 36 and 45 μM for bovine erythrocyte and electric eel enzyme, respectively).{45085} It inhibits acetylcholine-induced contractions of isolated guinea pig ileum when used at a concentration of 2.5 μM.{45086}  

 

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SKU: 23865 - 50 mg Category:

Description

An antispasmodic agent; an inhibitor of AChE (Kis = 36 and 45 μM for bovine erythrocyte and electric eel enzyme, respectively); inhibits acetylcholine-induced contractions of isolated guinea pig ileum at 2.5 μM

Formal name: 2-[4-[2-(1-piperidinyl)ethoxy]benzoyl]-benzoic acid, methyl ester, monohydrochloride

Synonyms: 

Molecular weight: 403.9

CAS: 1248-42-6

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Small Molecule Inhibitors|Acetylcholine Turnover||Research Area|Neuroscience

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