An antimalarial agent; a bis-quinoline compound; inhibits the ex vivo growth of P. falciparum isolates from malaria-infected patients (IC50s = 11.8-217.3 nM)

Piperaquine – 100 mg

Brand:
Cayman
CAS:
4085-31-8
Storage:
-20
UN-No:
Non-Hazardous - /

Piperaquine is a bis-quinoline compound that inhibits the ex vivo growth of P. falciparum isolates from malaria-infected patients with IC50s ranging from 11.8-217.3 nM.{21232} Formulations containing piperaquine have been used in combination with artemisinin (Item No. 11816) for the treatment of malaria in HIV-1-positive populations.{28281,26531,26532}  

 

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Description

An antimalarial agent; a bis-quinoline compound; inhibits the ex vivo growth of P. falciparum isolates from malaria-infected patients (IC50s = 11.8-217.3 nM)

Formal name: 4,4′-(1,3-propanediyldi-4,1-piperazinediyl)bis[7-chloro-quinoline

Synonyms:  Piperaquinoline

Molecular weight: 535.5

CAS: 4085-31-8

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Antiparasitics|Antiprotozoals||Research Area|Immunology & Inflammation||Research Area|Infectious Disease|Parasitic Diseases|Malaria||Research Area|Infectious Disease|Viral Diseases|HIV & AIDS

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