A reversible antagonist of α-adrenergic receptors

Phentolamine (mesylate) – 500 mg

Brand:
Cayman
CAS:
65-28-1
Storage:
-20
UN-No:
Non-Hazardous - /

Phentolamine is a reversible antagonist of α-adrenergic receptors, non-specifically binding all α1- and α2-adrenoceptors with nanomolar affinities.{26301,23961,26302,25914} Formulations containing phentolamine have been used in the treatment of hypertensive emergencies, as well as chronic and emergent pain.  

 

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Description

A reversible antagonist of α-adrenergic receptors, non-specifically binding all α1- and α2-adrenoceptors with nanomolar affinities; rapidly and transiently increases local blood flow

Formal name: 3-[[(4,5-dihydro-1H-imidazol-2-yl)methyl](4-methylphenyl)amino]-phenol, monomethanesulfonate

Synonyms: 

Molecular weight: 377.5

CAS: 65-28-1

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Cardiovascular System|Cardiovascular Diseases|Hypertension||Research Area|Neuroscience|Pain Research

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