An oxytocin receptor antagonist (Ki = 9.5 nM); selective for the oxytocin receptor over the vasopressin receptors V1A and V2 (Kis = 1

PF-3274167 – 5 mg

Brand:
Cayman
CAS:
900510-03-4
Storage:
-20
UN-No:
Non-Hazardous - /

PF-3274167 is an oxytocin receptor antagonist (Ki = 9.5 nM).{43621} It is selective for the oxytocin receptor over the vasopressin receptors V1A and V2 (Kis = 1,120 and 10,000 nM, respectively).  

 

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SKU: 26189 - 5 mg Category:

Description

An oxytocin receptor antagonist (Ki = 9.5 nM); selective for the oxytocin receptor over the vasopressin receptors V1A and V2 (Kis = 1,120 and 10,000 nM, respectively)

Formal name: 5-[3-[3-(2-chloro-4-fluorophenoxy)-1-azetidinyl]-5-(methoxymethyl)-4H-1,2,4-triazol-4-yl]-2-methoxy-pyridine

Synonyms: 

Molecular weight: 419.8

CAS: 900510-03-4

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Endocrinology & Metabolism|Hormones & Receptors

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