A cyclodepsipeptide with anthelmintic activity; oral administration induces worm excretion in a chicken model of A. galli infection from 0.5-2 mg/kg; induces parasite clearance in jird models of H. contortus

PF-1022A – 5 mg

Brand:
Cayman
CAS:
133413-70-4
Storage:
-20
UN-No:
Non-Hazardous - /

PF-1022A is a cyclodepsipeptide fungal metabolite originally isolated from mycelia sterilia and has anthelmintic activity.{48890} Oral administration of PF-1022A (0.5-2 mg/kg) induces worm excretion in a chicken model of A. galli infection. It induces parasite clearance in jird models of H. contortus, O. ostertagi, or T. colubriformis infection (ED95s = 0.11, 0.33, and 0.11 mg/animal).{48891}  

 

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SKU: 29700 - 5 mg Category:

Description

A cyclodepsipeptide with anthelmintic activity; oral administration induces worm excretion in a chicken model of A. galli infection from 0.5-2 mg/kg; induces parasite clearance in jird models of H. contortus, O. ostertagi, or T. colubriformis infection (ED95s = 0.11, 0.33, and 0.11 mg/animal)

Formal name: cyclo[(αR)-α-hydroxybenzenepropanoyl-N-methyl-L-leucyl-(2R)-2-hydroxypropanoyl-N-methyl-L-leucyl-(αR)-α-hydroxybenzenepropanoyl-N-methyl-L-leucyl-(2R)-2-hydroxypropanoyl-N-methyl-L-leucyl]

Synonyms: 

Molecular weight: 949.2

CAS: 133413-70-4

Purity: ≥98%

Formulation: A crystalline solid

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