An orally active ACE inhibitor that effectively lowers blood pressure; metabolized to perindoprilat

Perindopril – 1 g

Brand:
Cayman
CAS:
82834-16-0
Storage:
-20
UN-No:
Non-Hazardous - /

Perindopril is an orally active angiotensin converting enzyme (ACE) inhibitor that effectively lowers blood pressure.{29639,29640} It is a prodrug that is metabolized to perindoprilat (Item No. 17574), a specific, competitive inhibitor of ACE (IC50 = 1.5-3.2 nM in vitro).{30687}  

 

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SKU: 20796 - Category:

Description

An orally active ACE inhibitor that effectively lowers blood pressure; metabolized to perindoprilat, a specific, competitive inhibitor of ACE (IC50 = 1.5-3.2 nM in vitro)

Formal name: (2S,3aS,7aS)-1-[(2S)-2-[[(1S)-1-(ethoxycarbonyl)butyl]amino]-1-oxopropyl]octahydro-1H-indole-2-carboxylic acid

Synonyms: 

Molecular weight: 368.5

CAS: 82834-16-0

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Small Molecule Inhibitors|Angiotensin-converting Enzyme||Research Area|Cardiovascular System|Cardiovascular Diseases|Hypertension

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