A histamine H1 receptor antagonist and a mast cell stabilizer that prevents the release of histamine; also blocks the release of substance P

Pemirolast (potassium salt) – 10 mg

Brand:
Cayman
CAS:
100299-08-9
Storage:
-20
UN-No:
Non-Hazardous - /

Pemirolast is a histamine H1 receptor antagonist and a mast cell stabilizer that prevents the release of histamine.{29107} It also blocks the release of substance P, neurokinin A, and calcitonin gene-related peptide from sensory nerves.{29108} Pemirolast has been used for the treatment of allergic conjunctivitis.{29106}  

 

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Description

A histamine H1 receptor antagonist and a mast cell stabilizer that prevents the release of histamine; also blocks the release of substance P, neurokinin A, and calcitonin gene-related peptide from sensory nerves

Formal name: 9-methyl-3-(2H-tetrazol-5-yl)-4H-pyrido[1,2-a]pyrimidin-4-one, monopotassium salt

Synonyms:  BMY 26517|TBX

Molecular weight: 266.3

CAS: 100299-08-9

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Immunology & Inflammation|Allergy||Research Area|Immunology & Inflammation|Innate Immunity||Research Area|Neuroscience|Ophthalmology

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