An opium alkaloid that is structurally and pharmacologically distinct from opiates; inhibits phosphodiesterase activity (IC50 = 13 μM) to increase cellular cAMP levels and alter cellular function; reduces heart and brain vasospasm and has been used to treat erectile dysfunction

Papaverine – 100 mg

Brand:
Cayman
CAS:
58-74-2
Storage:
-20
UN-No:
Non-Hazardous - /

Papaverine is an opium alkaloid that is structurally and pharmacologically distinct from opiates. At the cellular level, papaverine inhibits phosphodiesterase activity (IC50 = 13 μM).{16575} Through this action, it increases cellular cAMP levels and alters cellular function. It has been shown to reduce arterial and cerebral vasospasm and has been used to treat erectile dysfunction.{16574,16576,22,705} Papaverine is recommended as a potent nonselective phosphodiesterase inhibitor for in vitro and in vivo research purposes.  

 

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SKU: 10011133 - 100 mg Category:

Description

An opium alkaloid that is structurally and pharmacologically distinct from opiates; inhibits phosphodiesterase activity (IC50 = 13 μM) to increase cellular cAMP levels and alter cellular function; reduces heart and brain vasospasm and has been used to treat erectile dysfunction

Formal name: 1-[(3,4-dimethoxyphenyl)methyl]-6,7-dimethoxy isoquinoline

Synonyms:  NSC 136630

Molecular weight: 339.4

CAS: 58-74-2

Purity: ≥98%

Formulation: A crystalline solid

Application|Mass Spectrometry||Product Type|Biochemicals|Analytical Standards||Product Type|Biochemicals|Drugs of Abuse||Research Area|Forensic Chemistry & Toxicology|Sedatives & Muscle Relaxers

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