A fungal metabolite; inhibits HIV-1 integrase (IC50s = 350 and 268 µM for 3’-processing and strand transfer activity

Palitantin – 2.5 mg

Brand:
Cayman
CAS:
15265-28-8
Storage:
-20
UN-No:
- /

Palitantin is a fungal metabolite originally isolated from P. palitans.{39756} It inhibits HIV-1 integrase with IC50 values of 350 and 268 µM for 3’-processing and strand transfer activity, respectively.{39757} Palitantin has been used as a standard for dereplication of natural products.{41781}  

 

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SKU: 25208 - 2.5 mg Category:

Description

A fungal metabolite; inhibits HIV-1 integrase (IC50s = 350 and 268 µM for 3’-processing and strand transfer activity, respectively); has been used as a standard for dereplication of natural products

Formal name: (2R,3S,5R,6R)-rel-3-(1E,3E)-1,3-heptadien-1-yl-5,6-dihydroxy-2-(hydroxymethyl)-cyclohexanone

Synonyms:  ,NSC 246119,|(±)-Palitantin

Molecular weight: 254.3

CAS: 15265-28-8

Purity: ≥95%

Formulation: A solid

Product Type|Biochemicals|Antivirals|Integrase Inhibitors||Product Type|Biochemicals|Natural Products|Microbial Metabolites||Product Type|Biochemicals|Small Molecule Inhibitors|Nucleic Acid Turnover/Signaling||Research Area|Immunology & Inflammation||Research Area|Infectious Disease|Viral Diseases|HIV & AIDS

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