An irreversible inhibitor of serine proteases (Kis = 1.02

p-APMSF (hydrochloride) – 10 mg

Brand:
Cayman
CAS:
74938-88-8
Storage:
-20
UN-No:
Non-Hazardous - /

p-APMSF is an irreversible inhibitor of serine proteases with Ki values of 1.02, 1.18, 1.5, and 1.54 µM for bovine trypsin, human thrombin, bovine plasmin, and bovine Factor Xa, respectively.{25670} It is selective for these proteases over bovine chymotrypsin and acetylcholinesterase.  

 

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Description

An irreversible inhibitor of serine proteases (Kis = 1.02, 1.18, 1.5, and 1.54 µM for bovine trypsin, human thrombin, bovine plasmin, and bovine Factor Xa, respectively); selective for these proteases over bovine chymotrypsin and acetylcholinesterase

Formal name: 4-(aminoiminomethyl)-benzenemethanesulfonyl fluoride, monohydrochloride

Synonyms:  (p-Amidinophenyl)methanesulfonyl Fluoride|para-APMSF

Molecular weight: 252.7

CAS: 74938-88-8

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Small Molecule Inhibitors|Peptidases & Proteases||Research Area|Cell Biology|Proteolysis|Cytosolic & Secreted Proteases

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