A reversible inhibitor of Ca2+-independent PLA2; inhibits epinephrine-stimulated thromboxane production in human platelets

ONO-RS-082 – 100 mg

Brand:
Cayman
CAS:
99754-06-0
Storage:
-20
UN-No:
De Minimis - 3077 / 9

ONO-RS-082 is a reversible inhibitor of Ca2+-independent phospholipase A2.{32316} At 3.5 µM, it has been shown to inhibit epinephrine-stimulated thromboxane production in human platelets.{32316} ONO-RS-082 can also disrupt endosome tubule formation and maintenance of the Golgi complex.{9879,32317}  

 

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Description

A reversible inhibitor of Ca2+-independent PLA2; inhibits epinephrine-stimulated thromboxane production in human platelets

Formal name: 4-chloro-2-[[(2E)-1-oxo-3-(4-pentylphenyl)-2-propen-1-yl]amino]-benzoic acid

Synonyms: 

Molecular weight: 371.9

CAS: 99754-06-0

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Small Molecule Inhibitors|Phospholipases||Research Area|Cardiovascular System|Blood||Research Area|Cell Biology|Endomembrane System & Vesicular Trafficking||Research Area|Lipid Biochemistry|Glycerophospholipids|Phospholipases

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