A major active metabolite of metoprolol; formed by metabolism of metoprolol by CYP2D6 in vivo

O-Desmethyl Metoprolol – 5 mg

Brand:
Cayman
CAS:
62572-94-5
Storage:
-20
UN-No:
Non-Hazardous - /

O-Desmethyl metoprolol is the major active metabolite of the β1-adrenergic receptor blocker metoprolol (Item No. 15429 | 21165).{35205} It is formed by metabolism of metoprolol by the cytochrome P450 (CYP) isoform CYP2D6 in vivo.{35202}  

 

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Description

A major active metabolite of metoprolol; formed by metabolism of metoprolol by CYP2D6 in vivo

Formal name: 4-[2-hydroxy-3-[(1-methylethyl)amino]propoxy]-benzeneethanol

Synonyms:  O-DMM|SL 80-0088

Molecular weight: 253.3

CAS: 62572-94-5

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Product Type|Biochemicals|Xenobiotic Metabolites||Research Area|Cardiovascular System|Cardiovascular Diseases||Research Area|Cardiovascular System|Heart|Arrhythmia||Research Area|Toxicology|Drug Metabolism|Cytochrome P450||Research Area|Toxicology|Drug Metabolism|Drug Metabolites

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