An analog of pyrovalerone that is characterized by the substitution of the methylphenyl group of pyrovalerone with a naphthyl group; potently inhibits dopamine

Naphyrone (hydrochloride) (exempt preparation) – 1 mg

Brand:
Cayman
CAS:
850352-11-3
Storage:
-20
UN-No:
De Minimis - 1230 / 3|6.1

Pyrovalerone is a psychoactive compound with stimulatory effects. It is a controlled drug that has been found as a contaminant in products sold as bath salts. Naphyrone (hydrochloride) is an analog of pyrovalerone that is characterized by the substitution of the methylphenyl group of pyrovalerone with a naphthyl group. Naphyrone potently inhibits dopamine, serotonin, and norepinephrine transporters (IC50 = 20, 33, and 136 nM, respectively).{18943} Naphyrone, like pyrovalerone, has been detected in bath salt-type products. This compound is intended for forensic and research purposes.  

 

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Description

An analog of pyrovalerone that is characterized by the substitution of the methylphenyl group of pyrovalerone with a naphthyl group; potently inhibits dopamine, serotonin, and norepinephrine transporters (IC50 = 20, 33, and 136 nM, respectively); intended for forensic and research purposes

Formal name: 1-(2-naphthalenyl)-2-(1-pyrrolidinyl)-1-pentanone, monohydrochloride

Synonyms:  Naphpyrovalerone|NRG-1|O-2482|β-Naphyrone

Molecular weight: 317.9

CAS: 850352-11-3

Purity: ≥97%

Formulation: A solution in methanol

Application|Mass Spectrometry||Product Type|Biochemicals|Drugs of Abuse||Research Area|Forensic Chemistry & Toxicology|Stimulants|Cathinones

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