An active metabolite of zolmitriptan; an agonist of 5-HT1B receptors; induces contraction of isolated human cerebral arteries (EC50 = 100 nM)

N-desmethyl Zolmitriptan – 5 mg

Brand:
Cayman
CAS:
139264-35-0
Storage:
-20
UN-No:
Non-Hazardous - /

N-desmethyl Zolmitriptan (DZT) is an active metabolite of the serotonin (5-HT) receptor subtype 5-HT1B and 5-HT1D agonist zolmitriptan (Item No. 15871).{43950} DZT is an agonist of 5-HT1B receptors that induces contraction of isolated human cerebral arteries (EC50 = 100 nM).{43951}  

 

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SKU: 28058 - 5 mg Category:

Description

An active metabolite of zolmitriptan; an agonist of 5-HT1B receptors; induces contraction of isolated human cerebral arteries (EC50 = 100 nM)

Formal name: 4(S)-[[3-[2-(methylamino)ethyl]-1H-indol-5-yl]methyl]-2-oxazolidinone

Synonyms:  183C91|DZT

Molecular weight: 273.3

CAS: 139264-35-0

Purity: ≥95%

Formulation: A solid

Product Type|Biochemicals|Receptor Pharmacology|Agonists||Product Type|Biochemicals|Xenobiotic Metabolites||Research Area|Neuroscience|Pain Research||Research Area|Toxicology|Drug Metabolism|Drug Metabolites

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