A histamine metabolite; selectively inhibits sweet-almond β-glucosidase over yeast α-glucosidase in vitro (Kis = 0.035 and 20 mM

N-acetyl Histamine – 500 mg

Brand:
Cayman
CAS:
673-49-4
Storage:
-20
UN-No:
Non-Hazardous - /

N-acetyl Histamine is a histamine metabolite that is formed via acetyl-CoA-dependent N-acetylation of histamine by AANATL7 in D. melanogaster, polyamine N-acetyltransferase in F. hepatica, and the arylalkylamine N-acetyltransferases aaNAT2 and aaNAT5b in A. aegypti.{41784} It selectively inhibits sweet-almond β-glucosidase over yeast α-glucosidase in vitro (Kis = 0.035 and 20 mM, respectively).{41783} It also inhibits human glutaminyl cyclase (IC50 = 17 μM).{41785} N-acetyl Histamine has no effect on eosinophil activity and has been used as a negative control for histamine mediation of anaphylaxis.{41786}  

 

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SKU: 25118 - 500 mg Category:

Description

A histamine metabolite; selectively inhibits sweet-almond β-glucosidase over yeast α-glucosidase in vitro (Kis = 0.035 and 20 mM, respectively); inhibits human glutaminyl cyclase (IC50 = 17 μM); has been used as a negative control for histamine mediation of anaphylaxis

Formal name: N-[2-(1H-imidazol-5-yl)ethyl]-acetamide

Synonyms:  NSC 66356|Nω-Acetylhistamine

Molecular weight: 153.2

CAS: 673-49-4

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Small Molecule Inhibitors||Product Type|Biochemicals|Xenobiotic Metabolites

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