A positive allosteric modulator of nAChRs; enhances channel gating of the α3β2 nAChR subtype

Morantel (tartrate) – 1 g

Brand:
Cayman
CAS:
26155-31-7
Storage:
-20
UN-No:
Non-Hazardous - /

Morantel is a positive allosteric modulator of neuronal nicotinic acetylcholine receptors (nAChRs).{39211} It enhances channel gating of the α3β2 nAChR subtype by binding to non-canonical sites.{39210} Formulations containing morantel are used to treat nematode infections in livestock.{39209}  

 

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Description

A positive allosteric modulator of nAChRs; enhances channel gating of the α3β2 nAChR subtype

Formal name: 1,4,5,6-tetrahydro-1-methyl-2-[(2E)-2-(3-methyl-2-thienyl)ethenyl]-pyrimidine, 2R,3R-dihydroxybutanedioate

Synonyms:  CP 12,009-18|UK 2964-18

Molecular weight: 370.4

CAS: 26155-31-7

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Ion Channel Modulation|Activators||Research Area|Immunology & Inflammation||Research Area|Infectious Disease|Parasitic Diseases||Research Area|Neuroscience

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