A prodrug to mometasone

Mometasone Furoate – 250 mg

Brand:
Cayman
CAS:
83919-23-7
Storage:
-20
UN-No:
Non-Hazardous - /

Mometasone furoate is a prodrug to mometasone, a glucocorticoid receptor agonist.{33206} Like other corticosteroids, mometasone furoate suppresses allergic, inflammatory, and immune responses in various experimental models.{33597} Mometasone furoate has been shown to decrease NF-κB activity in a farnesoid X receptor-dependent manner.{33596}  

 

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Description

A prodrug to mometasone, a glucocorticoid receptor agonist; suppresses allergic, inflammatory, and immune responses in various experimental models

Formal name: 9,21-dichloro-17-[(2-furanylcarbonyl)oxy]-11β-hydroxy-16α-methyl-pregna-1,4-diene-3,20-dione

Synonyms:  SCH 32088

Molecular weight: 521.4

CAS: 83919-23-7

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Endocrinology & Metabolism|Bile Acids & Microbiome||Research Area|Endocrinology & Metabolism|Hormones & Receptors|FXRs & LXRs||Research Area|Endocrinology & Metabolism|Hormones & Receptors|Glucocorticoids & Mineralocorticoids||Research Area|Immunology & Inflammation|Allergy

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