A carbamate pesticide; inhibits AChE activity and is toxic to the western flower thrip (F. occidentalis; IC50 = 2.1 μM; LC50 = 3.26 ppm); toxic to the land snail M. obstructa (LD50 = 27.4 μg/snail) and the citrus mite A. pelekassi; reduces the seasonal percentages of cotton bolls infested with pink bollworm (P. gossypiella) to 4% when applied to cotton fields at 1.86 lb/acre; reduces damage to grapes by song birds when applied to vineyards at 2.5 lbs AI per 100 gal water per acre; is an ERα and ERβ agonist (EC20s = 19.87 and 20.24 μM

Methiocarb – 100 mg

Brand:
Cayman
CAS:
2032-65-7
Storage:
-20
UN-No:
- /

Methiocarb is a carbamate pesticide with insecticidal, molluscicidal, acaricidal, and bird repellant properties.{43317,43318,43319,43320,43323} It inhibits acetylcholinesterase (AChE) activity and is toxic to the western flower thrip (F. occidentalis; IC50 = 2.1 μM; LC50 = 3.26 ppm).{43318} Methiocarb is also toxic to the land snail M. obstructa (LD50 = 27.4 μg/snail) and the citrus mite A. pelekassi, inducing 94% mortality when used at a concentration of 0.5 ppm.{43317,43319} It reduces the seasonal percentages of cotton bolls infested with pink bollworm (P. gossypiella) to 4%, compared with 65% infestation in untreated controls, when applied to cotton fields at a concentration of 1.86 lb/acre.{43323} Methiocarb reduces damage to grapes by song birds when applied to vineyards at a concentration of 2.5 lbs AI per 100 gal water per acre.{43320} It is an estrogen receptor α (ERα) and ERβ agonist (EC20s = 19.87 and 20.24 μM, respectively) and an androgen receptor antagonist (IC50 = 13.89 μM) in cell-based reporter assays.{43321} It is toxic to juvenile rainbow trout (O. mykiss) and guppies (P. reticulata) with LC50 values of 0.8 and 1.48 mg/L, respectively, at 48 hours of exposure.{43322} Formulations containing methiocarb have been used in the agricultural control of pests.  

 

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SKU: 25627 - 100 mg Category:

Description

A carbamate pesticide; inhibits AChE activity and is toxic to the western flower thrip (F. occidentalis; IC50 = 2.1 μM; LC50 = 3.26 ppm); toxic to the land snail M. obstructa (LD50 = 27.4 μg/snail) and the citrus mite A. pelekassi; reduces the seasonal percentages of cotton bolls infested with pink bollworm (P. gossypiella) to 4% when applied to cotton fields at 1.86 lb/acre; reduces damage to grapes by song birds when applied to vineyards at 2.5 lbs AI per 100 gal water per acre; is an ERα and ERβ agonist (EC20s = 19.87 and 20.24 μM, respectively) and an androgen receptor antagonist (IC50 = 13.89 μM); toxic to juvenile rainbow trout (O. mykiss) and guppies (P. reticulata; LC50s = 0.8 and 1.48 mg/L, respectively)

Formal name: 3,5-dimethyl-4-(methylthio)-phenol, 1-(N-methylcarbamate)

Synonyms:  4-Methylthio-3,5-dimethylphenyl methylcarbamate|BAY 37344|Mercaptodimethur

Molecular weight: 225.3

CAS: 2032-65-7

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Pesticides|Acaricides||Product Type|Biochemicals|Pesticides|Insecticides||Product Type|Biochemicals|Receptor Pharmacology|Agonists||Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Product Type|Biochemicals|Small Molecule Inhibitors|MMPs||Research Area|Cell Biology||Research Area|Endocrinology & Metabolism|Hormones & Receptors||Research Area|Endocrinology & Metabolism|Reproductive Biology||Research Area|Neuroscience||Research Area|Toxicology|Environmental|Agriculture||Research Area|Toxicology|Environmental|Aquatic Systems||Research Area|Toxicology|Environmental|Endocrine Disruption

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