An analog of LTB4 that binds to the BLT1 and BLT2 receptors with Ki values of 5.1 and 1

Leukotriene B4-3-aminopropylamide – 100 µg

Brand:
Cayman
CAS:
89596-43-0
Storage:
-20
UN-No:
De Minimis - 1170 / 3

The effects of leukotriene B4 (LTB4) are mediated by two receptors, BLT1 and BLT2.{4425,8280} LTB4-3-aminopropylamide is an analog of LTB4 that exhibits potent and selective binding to the BLT1 receptor, having Ki values of 5.1 and 1,227 nM at BLT1 and BLT2, respectively.{8743}  

 

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SKU: 20114 - Category:

Description

An analog of LTB4 that binds to the BLT1 and BLT2 receptors with Ki values of 5.1 and 1,227 nM, respectively

Formal name: N-(3-aminopropyl)-5S,12R-dihydroxy-6Z,8E,10E,14Z-eicosatetraenamide

Synonyms:  LTB4-3-aminopropylamide

Molecular weight: 392.6

CAS: 89596-43-0

Purity: ≥95%

Formulation: A solution in ethanol

Product Type|Biochemicals|Lipids|Leukotrienes||Product Type|Biochemicals|Receptor Pharmacology||Research Area|Immunology & Inflammation||Research Area|Lipid Biochemistry|Lipoxygenase Pathways

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