An aminoalkylindole that acts as a CB receptor ligand

JWH 200 (exempt preparation) – 5 mg

Brand:
Cayman
CAS:
103610-04-4
Storage:
-20
UN-No:
De Minimis - 1648 / 3

JWH 200 is an aminoalkylindole that acts as a cannabinoid (CB) receptor ligand. It binds to the CB1 receptor with high-affinity (IC50 = 7.8-42 nM).{16961,16684} The effects of JWH 200 in locomotor activity, tail-flick latency, hypothermia and ring-immobility tests are comparable or superior to Δ9-THC or WIN 55,212.{16963} It potently inhibits the contraction of electrically-stimulated murine vas deferens (IC50 = 3.7-6.0 nM).{16960,16962}  

 

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Description

An aminoalkylindole that acts as a CB receptor ligand, binding the CB1 receptor with high affinity (IC50 = 7.8-42 nM)

Formal name: [1-[2-(4-morpholinyl)ethyl]-1H-indol-3-yl]-1-naphthalenyl-methanone

Synonyms: 

Molecular weight: 384.5

CAS: 103610-04-4

Purity: ≥98%

Formulation: A solution in acetonitrile

Application|Mass Spectrometry||Product Type|Biochemicals|Analytical Standards||Product Type|Biochemicals|Drugs of Abuse||Research Area|Forensic Chemistry & Toxicology|Cannabinoids|Synthetic Cannabinoids

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