A naphthoyl pyrrole cannabimimetic which activates the CB1 receptor (EC50 = 30.5 nM for rat

JWH 030 – 10 mg

Brand:
Cayman
CAS:
162934-73-8
Storage:
-20
UN-No:
De Minimis - 1230 / 3|6.1

JWH 030 is a naphthoyl pyrrole cannabimimetic which activates the CB1 receptor (EC50 = 30.5 nM for rat, Ki = 87 nM for mouse) better than CB2 (EC50 = 552 nM for human CB2).{11496,20068} JWH 030 is quite potent in vivo in the mouse spontaneous activity and tail flick (antinociception) assays (ED50 = 26.8 μM/kg).{20068} It also dose-dependently inhibits electrically-induced contractions of the mouse vas deferens (IC50 = 3.38 nM).{20069} This product is intended for forensic or research purposes.  

 

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SKU: 10831 - 10 mg Category:

Description

A naphthoyl pyrrole cannabimimetic which activates the CB1 receptor (EC50 = 30.5 nM for rat, Ki = 87 nM for mouse) better than CB2 (EC50 = 552 nM for human CB2); potent in vivo in the mouse spontaneous activity and tail flick (antinociception) assays (ED50 = 26.8 μM/kg)

Formal name: 1-naphthalenyl(1-pentyl-1H-pyrrol-3-yl)-methanone

Synonyms: 

Molecular weight: 291.4

CAS: 162934-73-8

Purity: ≥98%

Formulation: A solution in methanol

Product Type|Biochemicals|Drugs of Abuse||Research Area|Forensic Chemistry & Toxicology|Cannabinoids|Synthetic Cannabinoids

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