An irreversible FAAH inhibitor of the carbamate class with an IC50 value of 14 nM for the human recombinant enzyme when tested using radiolabeled oleamide as the substrate

JP83 – 10 mg

Brand:
Cayman
CAS:
887264-44-0
Storage:
-20
UN-No:
Non-Hazardous - /

The enzyme fatty acyl amide hydrolase (FAAH) is widely expressed in brain and other tissues, and is capable of hydrolyzing anandamide (AEA) and other simple esters and amides with long unsaturated acyl chains.{3110} JP83 is an irreversible fatty acyl amide hydrolase (FAAH) inhibitor of the carbamate class with an IC50 of 14 nM for the human recombinant enzyme when tested using radiolabeled oleamide as the substrate.{14130}  

 

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SKU: 10008660 - 10 mg Category:

Description

An irreversible FAAH inhibitor of the carbamate class with an IC50 value of 14 nM for the human recombinant enzyme when tested using radiolabeled oleamide as the substrate

Formal name: 3′-carbamoyl-biphenyl-3-yl-hexylphenylcarbamate

Synonyms: 

Molecular weight: 416.5

CAS: 887264-44-0

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Small Molecule Inhibitors|Fatty Acid Metabolism||Research Area|Lipid Biochemistry|Endocannabinoid/Endocannabinoid-like||Research Area|Neuroscience|Cannabinoid Research|Endocannabinoids

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