A metabolite of iloperidone; binds to 5-HT2A receptors and α1-

Iloperidone metabolite P95 – 1 mg

Brand:
Cayman
CAS:
475110-48-6
Storage:
-20
UN-No:
Non-Hazardous - /

Iloperidone metabolite P95 is a metabolite of the atypical antipsychotic iloperidone (Item No. 22957).{43847,43848} It binds to the serotonin (5-HT) receptor subtype 5-HT2A and α1-, α2B-, and α2C-adrenergic receptors with mean Ki values of 7.08, 21.38, 83.18, and 47.86 nM, respectively, but does not cross the blood-brain barrier.{43847}  

 

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SKU: 27807 - 1 mg Category:

Description

A metabolite of iloperidone; binds to 5-HT2A receptors and α1-, α2B- and α2C-adrenergic receptors (mean Kis = 7.08, 21.38, 83.18, and 47.86 nM, respectively); does not cross the blood-brain barrier

Formal name: 4-[3-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]propoxy]-3-methoxy-benzoic acid

Synonyms:  P95-12113

Molecular weight: 428.5

CAS: 475110-48-6

Purity: ≥98%

Formulation: A solid

Product Type|Biochemicals|Receptor Pharmacology||Product Type|Biochemicals|Xenobiotic Metabolites||Research Area|Neuroscience|Behavioral Neuroscience|Anxiety||Research Area|Neuroscience|Behavioral Neuroscience|Schizophrenia & Psychosis||Research Area|Toxicology|Drug Metabolism|Drug Metabolites

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