A selective adenosine A3 receptor agonist (Kis = 1.1

HEMADO – 10 mg

Brand:
Cayman
CAS:
403842-38-6
Storage:
-20
UN-No:
Non-Hazardous - /

HEMADO is a selective agonist of the adenosine A3 receptor (Kis = 1.1, 327, and 1,230 nM for A3, A1, and A2A receptors, respectively).{35294} HEMADO reduces release of lactate dehydrogenase (LDH) and creatine kinase-MB (CK-MB) from myocardium in isolated rat hearts subjected to ischemia-reperfusion injury.{35295}  

 

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Description

A selective adenosine A3 receptor agonist (Kis = 1.1, 327, and 1,230 nM for A3, A1, and A2A receptors, respectively); reduces release of LDH and CK-MB from myocardium in isolated rat hearts subjected to ischemia-reperfusion injury

Formal name: 2-(1-hexyn-1-yl)-N-methyl-adenosine

Synonyms: 

Molecular weight: 361.4

CAS: 403842-38-6

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Cardiovascular System|Cardiovascular Diseases|Myocardial Infarction

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