A non-selective protein kinase inhibitor (IC50s = 20

H-7 (hydrochloride) – 5 mg

Brand:
Cayman
CAS:
108930-17-2
Storage:
-20
UN-No:
Non-Hazardous - /

H-7 is a non-selective inhibitor of protein kinases (PKs; IC50s = 20, 36, 7, and 420 μM for PKC, A, G, and M, respectively).{38451} It has been widely used to characterize the functional roles of PKC in a multitude of cellular processes.{38451,38450}  

 

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Description

A non-selective protein kinase inhibitor (IC50s = 20, 36, 7, and 420 μM for PKC, A, G, and M, respectively); has been widely used to characterize the functional roles of PKC in a multitude of cellular processes,

Formal name: 5-[(2-methyl-1-piperazinyl)sulfonyl]-isoquinoline, dihydrochloride

Synonyms: 

Molecular weight: 364.3

CAS: 108930-17-2

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Kinase Inhibitors|PKA||Product Type|Biochemicals|Kinase Inhibitors|PKC||Product Type|Biochemicals|Kinase Inhibitors|PKD & PKG||Product Type|Biochemicals|Small Molecule Inhibitors|Kinases||Research Area|Cell Biology|Cell Signaling

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