An α2-adrenergic receptor agonist (effective concentrations 10-100 nM) with hypotensive effects; competes for imidazoline I2-binding sites in brown adipose tissue (Ki = 97 nM)

Guanabenz (hydrochloride) – 100 mg

Brand:
Cayman
CAS:
23113-43-1
Storage:
-20
UN-No:
Non-Hazardous - /

Guanabenz is an α2-adrenergic receptor agonist (effective concentrations 10-100 nM) with hypotensive effects.{20036}{20037} It also competes for imidazoline I2-binding sites in brown adipose tissue (Ki = 97 nM).{20035}  

 

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SKU: 10851 - 100 mg Category:

Description

An α2-adrenergic receptor agonist (effective concentrations 10-100 nM) with hypotensive effects; competes for imidazoline I2-binding sites in brown adipose tissue (Ki = 97 nM)

Formal name: 2-[(2,6-dichlorophenyl)methylene]-hydrazinecarboximidamide, monohydrochloride

Synonyms:  Wytensin

Molecular weight: 267.5

CAS: 23113-43-1

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Cardiovascular System|Vasculature|Vasodilation||Research Area|Neuroscience

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