A tropic hormone and agonist of GNRHR (Ki = 13 nM in CHO cells expressing the human receptor); stimulates LH and FSH release from rat anterior pituitary cultures (0.1 μg); stimulates LH release from bovine anterior pituitary cultures (1 μM); induces ovulation in rats pretreated with fluphenazine (ED50 = 610.3 ng/kg)

Gonadorelin (acetate) – 5 mg

Brand:
Cayman
CAS:
34973-08-5
Storage:
-20
UN-No:
Non-Hazardous - /

Gonadorelin is a tropic hormone and agonist of the gonadotropin-releasing hormone receptor (GNRHR; Ki = 13 nM in CHO cells expressing the human receptor).{36464} It stimulates luteinizing hormone (LH) and follicle-stimulating hormone (FSH) release from rat anterior pituitary cultures when administered at a dose of 0.1 μg.{40777} It also stimulates LH release from bovine anterior pituitary cultures at a concentration of 1 μM.{40778} In vivo, gonadorelin induces ovulation in rats pretreated with fluphenazine (Item No. 23555; ED50 = 610.3 ng/kg).{40779} Formulations containing gonadorelin have been used as diagnostic agents to assess pituitary gland function.  

 

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SKU: 24240 - 5 mg Category:

Description

A tropic hormone and agonist of GNRHR (Ki = 13 nM in CHO cells expressing the human receptor); stimulates LH and FSH release from rat anterior pituitary cultures (0.1 μg); stimulates LH release from bovine anterior pituitary cultures (1 μM); induces ovulation in rats pretreated with fluphenazine (ED50 = 610.3 ng/kg)

Formal name: luteinizing hormone-releasing factor (swine), acetate

Synonyms: 

Molecular weight: 1,182.30

CAS: 34973-08-5

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Peptides|Neuropeptides||Product Type|Biochemicals|Peptides|Peptide Hormones||Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Endocrinology & Metabolism|Hormones & Receptors||Research Area|Endocrinology & Metabolism|Reproductive Biology

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