A selective PAF receptor antagonist (IC50 = 37.6 μM); increases lipolysis and inhibits adipogenesis in adipocytes via the activated AMPK pathway

Ginkgolide C – 1 mg

Brand:
Cayman
CAS:
15291-76-6
Storage:
-20
UN-No:
Non-Hazardous - /

Ginkgolide C is a flavone first extracted from G. biloba leaves with multiple reported biological functions. It has been identified as a selective platelet activating factor receptor antagonist (IC50 = 37.6 μM).{6653} Ginkgolide C has also been shown to increase lipolysis and to inhibit adipogenesis in adipocytes via the activated AMPK pathway.{31746}  

 

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Description

A selective PAF receptor antagonist (IC50 = 37.6 μM); increases lipolysis and inhibits adipogenesis in adipocytes via the activated AMPK pathway

Formal name: (1S,2R,3S,3aS,4R,6aR,7aR,7bR,8S,10aS,11R,11aR)-3-(1,1-dimethylethyl)hexahydro-2,4,7b,11-tetrahydroxy-8-methyl-9H-1,7a-(epoxymethano)-1H,6aH-cyclopenta[c]furo[2,3-b]furo[3′,2′:3,4]cyclopenta[1,2-d]furan-5,9,12(4H)-trione

Synonyms:  1,7-dihydroxy Ginkgolide A|BN 52022

Molecular weight: 440.4

CAS: 15291-76-6

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Natural Products|Flavonoids||Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Endocrinology & Metabolism|Metabolic Diseases|Obesity

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