A synthetic progestin; binds to progesterone and androgen receptors (EC50s = 23 and 23.1 nM

Ethisterone – 1 g

Brand:
Cayman
CAS:
434-03-7
Storage:
-20
UN-No:
Non-Hazardous - /

Ethisterone is an orally bioavailable synthetic progestin and a derivative of testosterone (Item Nos. ISO60154 | 15645) that binds to progesterone and androgen receptors (EC50s = 23 and 23.1 nM, respectively, in yeast).{40099} Ethisterone (1 µM) downregulates progesterone receptors in MCF-7 cells.{40098}  

 

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SKU: 22893 - 1 g Category:

Description

A synthetic progestin; binds to progesterone and androgen receptors (EC50s = 23 and 23.1 nM, respectively, in yeast); downregulates progesterone receptors in MCF-7 cells at a concentration of 1 µM; a metabolite of danazol

Formal name: (17α)-hydroxy-pregn-4-en-20-yn-3-one

Synonyms: 

Molecular weight: 312.5

CAS: 434-03-7

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology||Research Area|Endocrinology & Metabolism|Hormones & Receptors|Androgens||Research Area|Endocrinology & Metabolism|Hormones & Receptors|Estrogens & Progestins

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