A decomposition product of the macrolide antibiotic

Erythromycin A enol ether – 5 mg

Brand:
Cayman
CAS:
33396-29-1
Storage:
-20
UN-No:
Non-Hazardous - /

Erythromycin A enol ether is a decomposition product of the macrolide antibiotic, erythromycin A (Item No. 16486).{25101} Erythromycin A enol ether does not retain the antibiotic properties of erythromycin A and has been identified as a β-turn mimic of the peptide hormone motilin, causing duodenal contractions and gastrointestinal distress.{28114} This compound has been used to determine the binding characteristics of ligands of the motilin receptor.{28114}  

 

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Description

A decomposition product of the macrolide antibiotic, erythromycin A that has been identified as a β-turn mimic of the peptide hormone motilin; used to determine the binding characteristics of ligands of the motilin receptor

Formal name: 8,9-didehydro-9-deoxo-6-deoxy-6,9-epoxy-erythromycin

Synonyms:  BRL 46357ER|EM-201

Molecular weight: 715.9

CAS: 33396-29-1

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Antibiotics|Macrolides||Product Type|Biochemicals|Peptides||Research Area|Endocrinology & Metabolism|Hormones & Receptors

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